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Valerian

Can I take valerian with my sleep medication?

By Dr. Paulette Y. Jones, DNP-L, RN · N&O LLC

Valerian and Sleep Medication: What Not to Combine

Valeriana officinalis

Valerian is the classic sleep herb, and it is a good one. It is also one of the clearest examples of an herb that should not be stacked on top of a prescription that does the same job. Here is what the studies found and the rule I give every customer.

What it is

Valerian is the root of a flowering plant native to Europe and Asia, used for sleep and nervous tension since ancient Greece. Its active compounds — valerenic acid and related valepotriates — increase the availability of GABA, the brain's main calming neurotransmitter, which is the same system that benzodiazepines and Z-drugs act on. Unlike those drugs it is not habit-forming, and it usually needs a couple of weeks of nightly use to show its full effect.

What the research has looked at

Doses used in research

Most trials used 300–600 mg of standardized root extract (0.8% valerenic acid) taken 30 minutes to 2 hours before bed, nightly, for at least two weeks. Evening Calm & Sleep uses 400 mg taken 2–3 hours before bed.

Interactions and cautions

Valerian adds to the effect of anything else that works on GABA: benzodiazepines, zolpidem and similar sleep drugs, barbiturates, opioids, sedating antihistamines, and alcohol. Combining them can cause excessive sedation and impaired breathing in the worst case. Do not drive after an evening dose. Rare liver reactions have been reported. Stop two weeks before surgery, because it can interact with anesthesia.

Drug / conditionSeverityWhyWhat to do
Benzodiazepines, barbiturates, Z-drugs, opioids, alcohol, antihistaminesMAJORAdditive CNS depressionDo not combine; no driving
AnesthesiaMODERATEProlonged sedation; withdrawal-like symptomsStop 2 weeks pre-surgery
CYP3A4 substratesMINORWeak inhibitionMonitor
Hepatotoxic drugs / liver diseaseMINORRare hepatotoxicity reportsMonitor
Loperamide, St. John's Wort, fluoxetineMINORCase reports of delirium/serotonergic effectsCaution
Who should not take it without a provider's approval: Anyone taking prescription sleep medication, benzodiazepines, or opioids without provider approval; alcohol on the same evening; pregnancy and nursing; two weeks before surgery; children.

Where we use it

Valerian extract 400 mg is in Evening Calm & Sleep, together with passionflower, L-theanine, lemon balm, magnolia bark, and ashwagandha. It is not in any other N&O LLC formula.

Dr. Paulette Y. Jones holds a Doctor of Nursing Practice in Leadership (DNP-L) and is a Registered Nurse with nearly thirty years of clinical experience. She is the founder and formulator of N&O LLC. This article is for education only and is not medical advice. *These statements have not been evaluated by the Food and Drug Administration. N&O LLC products are not intended to diagnose, treat, cure, or prevent any disease. Always consult your healthcare provider before starting, stopping, or combining any supplement with a medication.

Selected peer-reviewed references

Peer-reviewed journal sources supporting this article, prioritizing systematic reviews, meta-analyses, and randomized trials from the past five years. Current as of September 2026.

About the Formulator. Dr. Paulette Y. Jones holds a Doctor of Nursing Practice (DNP) with a specialization in Nursing Leadership (DNP-L) and is a Registered Nurse (RN). Dr. Jones is not a medical doctor (MD or DO), is not a nurse practitioner (NP or APRN), and is not a licensed independent prescriber. She does not hold prescriptive authority and does not practice medicine. In connection with N&O LLC, Dr. Jones acts solely as a product formulator, researcher, and wellness entrepreneur. Nothing on this website, on N&O LLC packaging, or in any communication from N&O LLC constitutes medical advice, diagnosis, or treatment, and no provider–patient relationship is created by purchasing or using any N&O LLC product.

Consult Your Provider First. Before taking any N&O LLC supplement, powder, capsule, or tea, consult your own primary care provider, prescribing clinician, or pharmacist — especially if you are pregnant, nursing, or trying to conceive; under 18; taking any prescription medication (including blood thinners, diabetes, blood pressure or heart medication, antidepressants or other psychiatric medication, thyroid or seizure medication, immunosuppressants, or disease-modifying therapies); living with a diagnosed medical condition; or scheduled for surgery. Bring the full ingredient list to that conversation. Your provider, not N&O LLC, should decide whether a product is appropriate for you.

Regulatory Statement. *These statements have not been evaluated by the U.S. Food and Drug Administration. N&O LLC products are dietary supplements and are not intended to diagnose, treat, cure, or prevent any disease. Dietary supplements are not a substitute for prescribed medication, and no N&O LLC product should be used to replace, reduce, or discontinue any medication without the direction of the prescribing provider. Product and protocol names (including “Shield,” “Guardian,” “Protect,” and similar words) are brand names describing intended wellness support and do not represent claims of medical efficacy. Interaction information is compiled from published literature, is not exhaustive, and should be re-verified with a professional before being relied upon. If you experience an unexpected symptom, stop use and contact your provider.